4-Acylamino-and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists
Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
Synthesis, in vitro biological evaluation and structure-activity relationships of 4-acylamino-and 4-ureidobenzamides as novel hMCH1R-antagonists are disclosed. The nature of the amine side chains could be varied considerably in contrast to the central benzamide scaffold and aromatic substituents.
Originalsprog | Engelsk |
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Tidsskrift | Bioorganic & Medicinal Chemistry Letters |
Vol/bind | 14 |
Udgave nummer | 20 |
Sider (fra-til) | 5075-5080 |
Antal sider | 6 |
ISSN | 0960-894X |
DOI | |
Status | Udgivet - 18 okt. 2004 |
ID: 189159527